Abstract
3-Hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles were discovered as potent in vitro MEK1 inhibitors.
MeSH terms
-
Drug Design
-
Enzyme Inhibitors / pharmacology*
-
MAP Kinase Kinase 1 / antagonists & inhibitors*
-
Thiazoles / pharmacology*
Substances
-
Enzyme Inhibitors
-
Thiazoles
-
MAP Kinase Kinase 1